1 |
10281 |
inhibitor |
10281 |
250.00 |
|
10281 |
2 |
138114219 |
inhibitor |
Control to be added |
360.00 |
|
To be Added |
3 |
4wxr-3zw |
Control |
{6-(3,5-diaminophenyl)-1-[4-(propan-2-yl)benzyl]-1H-indol-3-yl}acetic acid |
413.51 |
|
CC(C)c1ccc(Cn2cc(CC(O)=O)c3ccc(cc23)c4cc(N)cc(N)c4)cc1 |
4 |
5Qj0_j6d |
Control |
5QJ0_J6D |
627.68 |
|
CCN(c1cc2oc(c3ccc(F)cc3)c(C(=O)NC)c2cc1c4cccc(c4)C(=O)NC5(CC5)c6ncccn6)[S](C)(=O)=O |
5 |
637511 |
637511 |
637511 |
250.00 |
|
637511 |
6 |
6piv_olj |
Control |
|
54.00 |
|
to add1 |
7 |
DB00006 |
approved; investigational |
Bivalirudin |
2180.29 |
|
CC[C@H](C)[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC1=CC=CC=C1)NC(=O)[C@H](CC(O)=O)NC(=O)CNC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)CNC(=O)CNC(=O)CNC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H]1CCCN1C(=O)[C@H](N)CC1=CC=CC=C1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC1=CC=C(O)C=C1)C(=O)N[C@@H](CC(C)C)C(O)=O |
8 |
DB00007 |
approved; investigational |
Leuprolide |
1209.40 |
|
CCNC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](CC1=CC=C(O)C=C1)NC(=O)[C@H](CO)NC(=O)[C@H](CC1=CNC2=C1C=CC=C2)NC(=O)[C@H](CC1=CNC=N1)NC(=O)[C@@H]1CCC(=O)N1 |
9 |
DB00014 |
approved |
Goserelin |
1269.41 |
|
CC(C)C[C@H](NC(=O)[C@@H](COC(C)(C)C)NC(=O)[C@H](CC1=CC=C(O)C=C1)NC(=O)[C@H](CO)NC(=O)[C@H](CC1=CNC2=CC=CC=C12)NC(=O)[C@H](CC1=CN=CN1)NC(=O)[C@@H]1CCC(=O)N1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N1CCC[C@H]1C(=O)NNC(N)=O |
10 |
DB00027 |
approved |
Gramicidin D |
1811.25 |
|
CC(C)C[C@@H](NC(=O)CNC(=O)[C@@H](NC=O)C(C)C)C(=O)N[C@@H](C)C(=O)N[C@H](C(C)C)C(=O)N[C@@H](C(C)C)C(=O)N[C@H](C(C)C)C(=O)N[C@@H](CC1=CNC2=C1C=CC=C2)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](CC1=CNC2=C1C=CC=C2)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](CC1=CNC2=C1C=CC=C2)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](CC1=CNC2=C1C=CC=C2)C(=O)NCCO |
11 |
DB00035 |
approved |
Desmopressin |
1069.22 |
|
NC(=O)CC[C@@H]1NC(=O)[C@H](CC2=CC=CC=C2)NC(=O)[C@H](CC2=CC=C(O)C=C2)NC(=O)CCSSC[C@H](NC(=O)[C@H](CC(N)=O)NC1=O)C(=O)N1CCC[C@H]1C(=O)N[C@H](CCCNC(N)=N)C(=O)NCC(N)=O |
12 |
DB00050 |
approved; investigational |
Cetrorelix |
1431.04 |
|
CC(C)C[C@H](NC(=O)[C@@H](CCCNC(N)=O)NC(=O)[C@H](CC1=CC=C(O)C=C1)NC(=O)[C@H](CO)NC(=O)[C@@H](CC1=CN=CC=C1)NC(=O)[C@@H](CC1=CC=C(Cl)C=C1)NC(=O)[C@@H](CC1=CC2=CC=CC=C2C=C1)NC(C)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N1CCC[C@H]1C(=O)N[C@H](C)C(N)=O |
13 |
DB00080 |
approved; investigational |
Daptomycin |
1620.69 |
|
CCCCCCCCCC(=O)N[C@@H](CC1=CNC2=C1C=CC=C2)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@H]1[C@@H](C)OC(=O)[C@H](CC(=O)C2=C(N)C=CC=C2)NC(=O)[C@@H](NC(=O)[C@@H](CO)NC(=O)CNC(=O)[C@H](CC(O)=O)NC(=O)[C@@H](C)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CCCN)NC(=O)CNC1=O)[C@H](C)CC(O)=O |
14 |
DB00091 |
approved; investigational; vet_approved |
Cyclosporine |
1202.63 |
|
CC[C@@H]1NC(=O)[C@H]([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](NC(=O)[C@H](CC(C)C)N(C)C(=O)CN(C)C1=O)C(C)C |
15 |
DB00093 |
experimental |
Felypressin |
1040.22 |
|
NCCCC[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CSSC[C@H](N)C(=O)N[C@@H](CC2=CC=CC=C2)C(=O)N[C@@H](CC2=CC=CC=C2)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(N)=O)C(=O)N1)C(=O)NCC(N)=O |
16 |
DB00104 |
approved; investigational |
Octreotide |
1019.25 |
|
[H][C@]1(NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CC2=CNC3=C2C=CC=C3)NC(=O)[C@H](CC2=CC=CC=C2)NC(=O)[C@H](CSSC[C@H](NC1=O)C(=O)N[C@H](CO)[C@@H](C)O)NC(=O)[C@H](N)CC1=CC=CC=C1)[C@@H](C)O |
17 |
DB00106 |
approved; investigational; withdrawn |
Abarelix |
1416.09 |
|
CC(C)C[C@H](NC(=O)[C@@H](CC(N)=O)NC(=O)[C@H](CC1=CC=C(O)C=C1)N(C)C(=O)[C@H](CO)NC(=O)[C@@H](CC1=CN=CC=C1)NC(=O)[C@@H](CC1=CC=C(Cl)C=C1)NC(=O)[C@@H](CC1=CC2=C(C=CC=C2)C=C1)NC(C)=O)C(=O)N[C@@H](CCCCNC(C)C)C(=O)N1CCC[C@H]1C(=O)N[C@H](C)C(N)=O |
18 |
DB00114 |
approved; investigational; nutraceutical |
Pyridoxal phosphate |
247.14 |
|
CC1=NC=C(COP(O)(O)=O)C(C=O)=C1O |
19 |
DB00115 |
approved; nutraceutical |
Cyanocobalamin |
1355.37 |
|
C[C@H](CNC(=O)CC[C@]1(C)[C@@H](CC(N)=O)[C@H]2N=C1\C(C)=C1/N=C(/C=C3\N=C(\C(\C)=C4\[C@@H](CCC(N)=O)[C@](C)(CC(N)=O)[C@@]2(C)N4[Co+]C#N)[C@@](C)(CC(N)=O)[C@@H]3CCC(N)=O)C(C)(C)[C@@H]1CCC(N)=O)OP([O-])(=O)O[C@@H]1[C@@H](CO)O[C@@H]([C@@H]1O)N1C=NC2=C1C=C(C)C(C)=C2 |
20 |
DB00116 |
nutraceutical |
Tetrahydrofolic acid |
445.43 |
|
NC1=NC(=O)C2=C(NCC(CNC3=CC=C(C=C3)C(=O)N[C@@H](CCC(O)=O)C(O)=O)N2)N1 |
21 |
DB00117 |
investigational; nutraceutical |
Histidine |
155.16 |
|
N[C@@H](CC1=CNC=N1)C(O)=O |
22 |
DB00118 |
approved; investigational; nutraceutical |
Ademetionine |
398.44 |
|
[H][C@](N)(CC[S+](C)C[C@@]1([H])O[C@@]([H])(N2C=NC3=C(N)N=CN=C23)[C@]([H])(O)[C@]1([H])O)C([O-])=O |
23 |
DB00119 |
approved; investigational; nutraceutical |
Pyruvic acid |
88.06 |
|
CC(=O)C(O)=O |
24 |
DB00120 |
approved; investigational; nutraceutical |
Phenylalanine |
165.19 |
|
N[C@@H](CC1=CC=CC=C1)C(O)=O |
25 |
DB00121 |
approved; investigational; nutraceutical |
Biotin |
244.31 |
|
[H][C@]12CS[C@@H](CCCCC(O)=O)[C@@]1([H])NC(=O)N2 |
26 |
DB00122 |
approved; nutraceutical |
Choline |
104.17 |
|
C[N+](C)(C)CCO |
27 |
DB00123 |
approved; nutraceutical |
L-Lysine |
146.19 |
|
NCCCC[C@H](N)C(O)=O |
28 |
DB00125 |
investigational; nutraceutical |
Arginine |
174.20 |
|
N[C@@H](CCCNC(N)=N)C(O)=O |
29 |
DB00126 |
approved; nutraceutical |
Ascorbic acid |
176.12 |
|
[H][C@@]1(OC(=O)C(O)=C1O)[C@@H](O)CO |
30 |
DB00127 |
experimental; nutraceutical |
Spermine |
202.34 |
|
NCCCNCCCCNCCCN |
31 |
DB00128 |
approved; nutraceutical |
Aspartic acid |
133.10 |
|
N[C@@H](CC(O)=O)C(O)=O |
32 |
DB00129 |
approved; nutraceutical |
Ornithine |
132.16 |
|
NCCC[C@H](N)C(O)=O |
33 |
DB00130 |
approved; investigational; nutraceutical |
L-Glutamine |
146.14 |
|
N[C@@H](CCC(N)=O)C(O)=O |
34 |
DB00131 |
approved; investigational; nutraceutical |
Adenosine phosphate |
347.22 |
|
NC1=C2N=CN([C@@H]3O[C@H](COP(O)(O)=O)[C@@H](O)[C@H]3O)C2=NC=N1 |
35 |
DB00132 |
approved; investigational; nutraceutical |
alpha-Linolenic acid |
278.43 |
|
CC\C=C/C\C=C/C\C=C/CCCCCCCC(O)=O |
36 |
DB00133 |
investigational; nutraceutical |
Serine |
105.09 |
|
N[C@@H](CO)C(O)=O |
37 |
DB00134 |
approved; nutraceutical |
Methionine |
149.21 |
|
CSCC[C@H](N)C(O)=O |
38 |
DB00135 |
approved; investigational; nutraceutical |
Tyrosine |
181.19 |
|
N[C@@H](CC1=CC=C(O)C=C1)C(O)=O |
39 |
DB00136 |
approved; nutraceutical |
Calcitriol |
416.64 |
|
C[C@H](CCCC(C)(C)O)[C@@]1([H])CC[C@@]2([H])\C(CCC[C@]12C)=C\C=C1\C[C@@H](O)C[C@H](O)C1=C |
40 |
DB00137 |
approved; investigational; nutraceutical |
Lutein |
568.89 |
|
C\C(\C=C\C=C(/C)\C=C\[C@H]1C(C)=C[C@H](O)CC1(C)C)=C/C=C/C=C(\C)/C=C/C=C(\C)/C=C/C1=C(C)C[C@@H](O)CC1(C)C |
41 |
DB00138 |
approved; nutraceutical |
Cystine |
240.30 |
|
N[C@@H](CSSC[C@H](N)C(O)=O)C(O)=O |
42 |
DB00139 |
approved; nutraceutical |
Succinic acid |
118.09 |
|
OC(=O)CCC(O)=O |
43 |
DB00140 |
approved; investigational; nutraceutical; vet_approved |
Riboflavin |
376.36 |
|
CC1=C(C)C=C2N(C[C@H](O)[C@H](O)[C@H](O)CO)C3=NC(=O)NC(=O)C3=NC2=C1 |
44 |
DB00141 |
approved; investigational; nutraceutical |
N-Acetylglucosamine |
221.21 |
|
[H]C(=O)[C@H](NC(C)=O)[C@@H](O)[C@H](O)[C@H](O)CO |
45 |
DB00142 |
approved; nutraceutical |
Glutamic acid |
147.13 |
|
N[C@@H](CCC(O)=O)C(O)=O |
46 |
DB00143 |
approved; investigational; nutraceutical |
Glutathione |
307.32 |
|
N[C@@H](CCC(=O)N[C@@H](CS)C(=O)NCC(O)=O)C(O)=O |
47 |
DB00144 |
approved; investigational; nutraceutical |
Phosphatidyl serine |
385.30 |
|
CCCC(=O)O[C@H](COC(=O)CC)COP(O)(=O)OC[C@H](N)C(O)=O |
48 |
DB00145 |
approved; nutraceutical; vet_approved |
Glycine |
75.07 |
|
NCC(O)=O |
49 |
DB00146 |
approved; nutraceutical |
Calcifediol |
400.64 |
|
C[C@H](CCCC(C)(C)O)[C@@]1([H])CC[C@@]2([H])\C(CCC[C@]12C)=C\C=C1\C[C@@H](O)CCC1=C |
50 |
DB00147 |
experimental; nutraceutical |
Pyridoxal |
167.16 |
|
CC1=NC=C(CO)C(C=O)=C1O |
51 |
DB00148 |
approved; investigational; nutraceutical |
Creatine |
131.13 |
|
CN(CC(O)=O)C(N)=N |
52 |
DB00149 |
investigational; nutraceutical |
Leucine |
131.17 |
|
CC(C)C[C@H](N)C(O)=O |
53 |
DB00150 |
approved; nutraceutical; withdrawn |
Tryptophan |
204.23 |
|
N[C@@H](CC1=CNC2=C1C=CC=C2)C(O)=O |
54 |
DB00151 |
approved; nutraceutical |
Cysteine |
121.16 |
|
N[C@@H](CS)C(O)=O |
55 |
DB00152 |
approved; investigational; nutraceutical; vet_approved |
Thiamine |
265.36 |
|
CC1=C(CCO)SC=[N+]1CC1=CN=C(C)N=C1N |
56 |
DB00153 |
approved; nutraceutical |
Ergocalciferol |
396.65 |
|
CC(C)[C@@H](C)\C=C\[C@@H](C)[C@@]1([H])CC[C@@]2([H])\C(CCC[C@]12C)=C\C=C1\C[C@@H](O)CCC1=C |
57 |
DB00154 |
investigational; nutraceutical |
Dihomo-gamma-linolenic acid |
306.48 |
|
CCCCC\C=C/C\C=C/C\C=C/CCCCCCC(O)=O |
58 |
DB00155 |
approved; investigational; nutraceutical |
Citrulline |
175.19 |
|
N[C@@H](CCCNC(N)=O)C(O)=O |
59 |
DB00156 |
approved; nutraceutical |
Threonine |
119.12 |
|
C[C@@H](O)[C@H](N)C(O)=O |
60 |
DB00157 |
approved; nutraceutical |
NADH |
665.44 |
|
NC(=O)C1=CN(C=CC1)[C@@H]1O[C@H](CO[P@](O)(=O)O[P@](O)(=O)OC[C@H]2O[C@H]([C@H](O)[C@@H]2O)N2C=NC3=C(N)N=CN=C23)[C@@H](O)[C@H]1O |
61 |
DB00158 |
approved; nutraceutical; vet_approved |
Folic acid |
441.40 |
|
NC1=NC(=O)C2=NC(CNC3=CC=C(C=C3)C(=O)N[C@@H](CCC(O)=O)C(O)=O)=CN=C2N1 |
62 |
DB00159 |
approved; nutraceutical |
Icosapent |
302.45 |
|
CC\C=C/C\C=C/C\C=C/C\C=C/C\C=C/CCCC(O)=O |
63 |
DB00160 |
nutraceutical |
Alanine |
89.09 |
|
C[C@H](N)C(O)=O |
64 |
DB00161 |
approved; nutraceutical |
Valine |
117.15 |
|
CC(C)[C@H](N)C(O)=O |
65 |
DB00162 |
approved; nutraceutical; vet_approved |
Vitamin A |
286.45 |
|
C\C(=C/CO)\C=C\C=C(/C)\C=C\C1=C(C)CCCC1(C)C |
66 |
DB00163 |
approved; nutraceutical; vet_approved |
Vitamin E |
430.71 |
|
CC(C)CCC[C@@H](C)CCC[C@@H](C)CCC[C@]1(C)CCC2=C(O1)C(C)=C(C)C(O)=C2C |
67 |
DB00165 |
approved; investigational; nutraceutical; vet_approved |
Pyridoxine |
169.18 |
|
CC1=C(O)C(CO)=C(CO)C=N1 |
68 |
DB00166 |
approved; investigational; nutraceutical |
Lipoic acid |
206.33 |
|
OC(=O)CCCC[C@@H]1CCSS1 |
69 |
DB00167 |
investigational; nutraceutical |
Isoleucine |
131.17 |
|
CC[C@H](C)[C@H](N)C(O)=O |
70 |
DB00168 |
investigational; nutraceutical |
Aspartame |
294.30 |
|
COC(=O)[C@H](CC1=CC=CC=C1)NC(=O)[C@@H](N)CC(O)=O |
71 |
DB00169 |
approved; nutraceutical |
Cholecalciferol |
384.64 |
|
CC(C)CCC[C@@H](C)[C@@]1([H])CC[C@@]2([H])\C(CCC[C@]12C)=C\C=C1\C[C@@H](O)CCC1=C |
72 |
DB00170 |
approved; nutraceutical |
Menadione |
172.18 |
|
CC1=CC(=O)C2=CC=CC=C2C1=O |
73 |
DB00171 |
investigational; nutraceutical |
ATP |
507.18 |
|
NC1=NC=NC2=C1N=CN2[C@@H]1O[C@H](COP(O)(=O)OP(O)(=O)OP(O)(O)=O)[C@@H](O)[C@H]1O |
74 |
DB00172 |
nutraceutical |
Proline |
115.13 |
|
OC(=O)[C@@H]1CCCN1 |
75 |
DB00173 |
approved; nutraceutical |
Adenine |
135.13 |
|
NC1=C2NC=NC2=NC=N1 |
76 |
DB00174 |
approved; investigational; nutraceutical |
Asparagine |
132.12 |
|
N[C@@H](CC(N)=O)C(O)=O |
77 |
DB00175 |
approved |
Pravastatin |
424.53 |
|
[H][C@]12[C@H](C[C@H](O)C=C1C=C[C@H](C)[C@@H]2CC[C@@H](O)C[C@@H](O)CC(O)=O)OC(=O)[C@@H](C)CC |
78 |
DB00176 |
approved; investigational |
Fluvoxamine |
318.34 |
|
COCCCC\C(=N/OCCN)C1=CC=C(C=C1)C(F)(F)F |
79 |
DB00177 |
approved; investigational |
Valsartan |
435.52 |
|
CCCCC(=O)N(CC1=CC=C(C=C1)C1=CC=CC=C1C1=NNN=N1)[C@@H](C(C)C)C(O)=O |
80 |
DB00178 |
approved |
Ramipril |
416.51 |
|
[H][C@@]12CCC[C@]1([H])N([C@@H](C2)C(O)=O)C(=O)[C@H](C)N[C@@H](CCC1=CC=CC=C1)C(=O)OCC |
81 |
DB00179 |
approved; investigational |
Masoprocol |
302.37 |
|
C[C@@H](CC1=CC(O)=C(O)C=C1)[C@H](C)CC1=CC(O)=C(O)C=C1 |
82 |
DB00180 |
approved; investigational |
Flunisolide |
434.50 |
|
[H][C@@]12C[C@@]3([H])[C@]4([H])C[C@H](F)C5=CC(=O)C=C[C@]5(C)[C@@]4([H])[C@@H](O)C[C@]3(C)[C@@]1(OC(C)(C)O2)C(=O)CO |
83 |
DB00181 |
approved |
Baclofen |
213.66 |
|
NCC(CC(O)=O)C1=CC=C(Cl)C=C1 |
84 |
DB00182 |
approved; illicit; investigational |
Amphetamine |
135.21 |
|
CC(N)CC1=CC=CC=C1 |
85 |
DB00183 |
approved |
Pentagastrin |
767.90 |
|
CSCC[C@H](NC(=O)[C@H](CC1=CNC2=C1C=CC=C2)NC(=O)CCNC(=O)OC(C)(C)C)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CC1=CC=CC=C1)C(N)=O |
86 |
DB00184 |
approved |
Nicotine |
162.23 |
|
CN1CCC[C@H]1C1=CN=CC=C1 |
87 |
DB00185 |
approved |
Cevimeline |
199.31 |
|
CC1O[C@@]2(CS1)CN1CCC2CC1 |
88 |
DB00186 |
approved |
Lorazepam |
321.16 |
|
OC1N=C(C2=CC=CC=C2Cl)C2=C(NC1=O)C=CC(Cl)=C2 |
89 |
DB00187 |
approved |
Esmolol |
295.37 |
|
COC(=O)CCC1=CC=C(OCC(O)CNC(C)C)C=C1 |
90 |
DB00188 |
approved; investigational |
Bortezomib |
384.24 |
|
CC(C)C[C@H](NC(=O)[C@H](CC1=CC=CC=C1)NC(=O)C1=CN=CC=N1)B(O)O |
91 |
DB00189 |
approved; illicit; withdrawn |
Ethchlorvynol |
144.60 |
|
CCC(O)(\C=C\Cl)C#C |
92 |
DB00190 |
approved |
Carbidopa |
226.23 |
|
C[C@@](CC1=CC(O)=C(O)C=C1)(NN)C(O)=O |
93 |
DB00191 |
approved; illicit |
Phentermine |
149.23 |
|
CC(C)(N)CC1=CC=CC=C1 |
94 |
DB00192 |
approved |
Indecainide |
308.42 |
|
CC(C)NCCCC1(C(N)=O)C2=CC=CC=C2C2=CC=CC=C12 |
95 |
DB00193 |
approved; investigational |
Tramadol |
263.38 |
|
COC1=CC=CC(=C1)[C@@]1(O)CCCC[C@@H]1CN(C)C |
96 |
DB00194 |
approved; investigational |
Vidarabine |
267.24 |
|
NC1=NC=NC2=C1N=CN2[C@@H]1O[C@H](CO)[C@@H](O)[C@@H]1O |
97 |
DB00195 |
approved; investigational |
Betaxolol |
307.43 |
|
CC(C)NCC(O)COC1=CC=C(CCOCC2CC2)C=C1 |
98 |
DB00196 |
approved; investigational |
Fluconazole |
306.27 |
|
OC(CN1C=NC=N1)(CN1C=NC=N1)C1=C(F)C=C(F)C=C1 |
99 |
DB00197 |
approved; investigational; withdrawn |
Troglitazone |
441.54 |
|
CC1=C(C)C2=C(CCC(C)(COC3=CC=C(CC4SC(=O)NC4=O)C=C3)O2)C(C)=C1O |
100 |
DB00198 |
approved |
Oseltamivir |
312.40 |
|
CCOC(=O)C1=C[C@@H](OC(CC)CC)[C@H](NC(C)=O)[C@@H](N)C1 |